Ketoconazole K006-1G

产品介绍

Ketoconazole is an insoluble azole antimycotic compound that was discovered in 1976 (Janssen Pharmaceuticals) and patented in 1977.  It is a racemic mixture of the two enantiomers: levoketoconazole and dextroketoconazole.  It is a bioactive small molecule acting as a protein inhibitor, specifically inhibiting CYP3A5 involved in P-450-dependent steroid biosynthesis.  The compound has antineoplastic activity. 

Ketoconazole is soluble in DMSO, ethanol, chloroform, and methanol.

This product is considered a dangerous good. Quantities above 1 gram may be subject to additional shipping fees.